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Two-step synthesis of indeno[1,2-b]furazanopyrazines through combination of the SNH and Heck reactions. / Kvashnin, Yuriy a.; Belyaev, Danila v.; Kodess, Mikhail i. et al.
In: Mendeleev Communications, Vol. 33, No. 6, 01.11.2023, p. 753-755.

Research output: Contribution to journal › Article › peer-review

Harvard

Kvashnin, YA, Belyaev, DV, Kodess, MI, Ezhikova, MA, Rusinov, GL, Verbitskiy, EV & Charushin, VN 2023, 'Two-step synthesis of indeno[1,2-b]furazanopyrazines through combination of the SNH and Heck reactions', Mendeleev Communications, vol. 33, no. 6, pp. 753-755. https://doi.org/10.1016/j.mencom.2023.10.004

APA

Kvashnin, Y. A., Belyaev, D. V., Kodess, M. I., Ezhikova, M. A., Rusinov, G. L., Verbitskiy, E. V., & Charushin, V. N. (2023). Two-step synthesis of indeno[1,2-b]furazanopyrazines through combination of the SNH and Heck reactions. Mendeleev Communications, 33(6), 753-755. https://doi.org/10.1016/j.mencom.2023.10.004

Vancouver

Kvashnin YA, Belyaev DV, Kodess MI, Ezhikova MA, Rusinov GL, Verbitskiy EV et al. Two-step synthesis of indeno[1,2-b]furazanopyrazines through combination of the SNH and Heck reactions. Mendeleev Communications. 2023 Nov 1;33(6):753-755. doi: 10.1016/j.mencom.2023.10.004

Author

Kvashnin, Yuriy a. ; Belyaev, Danila v. ; Kodess, Mikhail i. et al. / Two-step synthesis of indeno[1,2-b]furazanopyrazines through combination of the SNH and Heck reactions. In: Mendeleev Communications. 2023 ; Vol. 33, No. 6. pp. 753-755.

BibTeX

@article{153b5b909e134712a685b7212d3295f6,
title = "Two-step synthesis of indeno[1,2-b]furazanopyrazines through combination of the SNH and Heck reactions",
abstract = "Enamines generated in situ from aliphatic amines and acetone react with 5-(2-bromophenyl)furazano[3,4-b]pyrazines via the nucleophilic substitution of hydrogen atom of the pyrazine ring. A representative of 9H-indeno[1,2-b]furazanopyrazin-9-ylidene ring system has been accessed by exploiting the intramolecular Heck cyclization of the obtained SNH-product. Several compounds derived from furazano[3,4-b]pyrazin-5-yl]prop-1-en-2-amines, proved to exhibit a bacteriostatic activity in vitro against Mycobacterium tuberculosis H37Rv.",
author = "Kvashnin, {Yuriy a.} and Belyaev, {Danila v.} and Kodess, {Mikhail i.} and Ezhikova, {Marina a.} and Rusinov, {Gennady l.} and Verbitskiy, {Egor v.} and Charushin, {Valery n.}",
year = "2023",
month = nov,
day = "1",
doi = "10.1016/j.mencom.2023.10.004",
language = "English",
volume = "33",
pages = "753--755",
journal = "Mendeleev Communications",
issn = "0959-9436",
publisher = "Royal Society of Chemistry",
number = "6",

}

RIS

TY - JOUR

T1 - Two-step synthesis of indeno[1,2-b]furazanopyrazines through combination of the SNH and Heck reactions

AU - Kvashnin, Yuriy a.

AU - Belyaev, Danila v.

AU - Kodess, Mikhail i.

AU - Ezhikova, Marina a.

AU - Rusinov, Gennady l.

AU - Verbitskiy, Egor v.

AU - Charushin, Valery n.

PY - 2023/11/1

Y1 - 2023/11/1

N2 - Enamines generated in situ from aliphatic amines and acetone react with 5-(2-bromophenyl)furazano[3,4-b]pyrazines via the nucleophilic substitution of hydrogen atom of the pyrazine ring. A representative of 9H-indeno[1,2-b]furazanopyrazin-9-ylidene ring system has been accessed by exploiting the intramolecular Heck cyclization of the obtained SNH-product. Several compounds derived from furazano[3,4-b]pyrazin-5-yl]prop-1-en-2-amines, proved to exhibit a bacteriostatic activity in vitro against Mycobacterium tuberculosis H37Rv.

AB - Enamines generated in situ from aliphatic amines and acetone react with 5-(2-bromophenyl)furazano[3,4-b]pyrazines via the nucleophilic substitution of hydrogen atom of the pyrazine ring. A representative of 9H-indeno[1,2-b]furazanopyrazin-9-ylidene ring system has been accessed by exploiting the intramolecular Heck cyclization of the obtained SNH-product. Several compounds derived from furazano[3,4-b]pyrazin-5-yl]prop-1-en-2-amines, proved to exhibit a bacteriostatic activity in vitro against Mycobacterium tuberculosis H37Rv.

UR - https://gateway.webofknowledge.com/gateway/Gateway.cgi?GWVersion=2&SrcAuth=tsmetrics&SrcApp=tsm_test&DestApp=WOS_CPL&DestLinkType=FullRecord&KeyUT=001128136700001

UR - http://www.scopus.com/inward/record.url?partnerID=8YFLogxK&scp=85183717530

U2 - 10.1016/j.mencom.2023.10.004

DO - 10.1016/j.mencom.2023.10.004

M3 - Article

VL - 33

SP - 753

EP - 755

JO - Mendeleev Communications

JF - Mendeleev Communications

SN - 0959-9436

IS - 6

ER -

ID: 50707657