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The design and Synthesis of 5-(morpholin-4-yl)-N'-sulfonyl-1,2,3-thiadiazole-4-amidines. / Dianova, Lidia N.; Beryozkina, Tetyana V.; Fan, Zhijin et al.
In: Chemistry of Heterocyclic Compounds, Vol. 58, No. 10, 01.09.2022, p. 543-546.

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Dianova LN, Beryozkina TV, Fan Z, Filimonov VO, Bakulev VA. The design and Synthesis of 5-(morpholin-4-yl)-N'-sulfonyl-1,2,3-thiadiazole-4-amidines. Chemistry of Heterocyclic Compounds. 2022 Sept 1;58(10):543-546. doi: 10.1007/s10593-022-03124-4

Author

Dianova, Lidia N. ; Beryozkina, Tetyana V. ; Fan, Zhijin et al. / The design and Synthesis of 5-(morpholin-4-yl)-N'-sulfonyl-1,2,3-thiadiazole-4-amidines. In: Chemistry of Heterocyclic Compounds. 2022 ; Vol. 58, No. 10. pp. 543-546.

BibTeX

@article{02986c4b7e8e4ad381e239ec01348541,
title = "The design and Synthesis of 5-(morpholin-4-yl)-N'-sulfonyl-1,2,3-thiadiazole-4-amidines",
abstract = "A strategy was proposed for the synthesis of 5-(morpholin-4-yl)-N'-sulfonyl-1,2,3-thiadiazole-4-imidamides, as well as previously unknown 2-thiocarbamoy lacetimidamides. Their reactions with arylsulfonyl azides were studied. In the case of reactions between dimorpholine derivatives of 2-thiocarbamoylacetimidamides and arylsulfonyl azides, diazo transfer did not occur. Instead, a new process was observed, producing the target molecules in one synthetic step via the formation of triazene intermediate and the elimination of ammonia.",
author = "Dianova, {Lidia N.} and Beryozkina, {Tetyana V.} and Zhijin Fan and Filimonov, {Valeriy O.} and Bakulev, {Vasiliy A.}",
note = "This study received financial support from the Russian Science Foundation within the framework of research project No. 18-13-00161. ",
year = "2022",
month = sep,
day = "1",
doi = "10.1007/s10593-022-03124-4",
language = "English",
volume = "58",
pages = "543--546",
journal = "Chemistry of Heterocyclic Compounds",
issn = "0009-3122",
publisher = "Springer Verlag",
number = "10",

}

RIS

TY - JOUR

T1 - The design and Synthesis of 5-(morpholin-4-yl)-N'-sulfonyl-1,2,3-thiadiazole-4-amidines

AU - Dianova, Lidia N.

AU - Beryozkina, Tetyana V.

AU - Fan, Zhijin

AU - Filimonov, Valeriy O.

AU - Bakulev, Vasiliy A.

N1 - This study received financial support from the Russian Science Foundation within the framework of research project No. 18-13-00161.

PY - 2022/9/1

Y1 - 2022/9/1

N2 - A strategy was proposed for the synthesis of 5-(morpholin-4-yl)-N'-sulfonyl-1,2,3-thiadiazole-4-imidamides, as well as previously unknown 2-thiocarbamoy lacetimidamides. Their reactions with arylsulfonyl azides were studied. In the case of reactions between dimorpholine derivatives of 2-thiocarbamoylacetimidamides and arylsulfonyl azides, diazo transfer did not occur. Instead, a new process was observed, producing the target molecules in one synthetic step via the formation of triazene intermediate and the elimination of ammonia.

AB - A strategy was proposed for the synthesis of 5-(morpholin-4-yl)-N'-sulfonyl-1,2,3-thiadiazole-4-imidamides, as well as previously unknown 2-thiocarbamoy lacetimidamides. Their reactions with arylsulfonyl azides were studied. In the case of reactions between dimorpholine derivatives of 2-thiocarbamoylacetimidamides and arylsulfonyl azides, diazo transfer did not occur. Instead, a new process was observed, producing the target molecules in one synthetic step via the formation of triazene intermediate and the elimination of ammonia.

UR - https://gateway.webofknowledge.com/gateway/Gateway.cgi?GWVersion=2&SrcAuth=tsmetrics&SrcApp=tsm_test&DestApp=WOS_CPL&DestLinkType=FullRecord&KeyUT=000877403400002

UR - http://www.scopus.com/inward/record.url?partnerID=8YFLogxK&scp=85146401451

U2 - 10.1007/s10593-022-03124-4

DO - 10.1007/s10593-022-03124-4

M3 - Article

VL - 58

SP - 543

EP - 546

JO - Chemistry of Heterocyclic Compounds

JF - Chemistry of Heterocyclic Compounds

SN - 0009-3122

IS - 10

ER -

ID: 33250508