1. 2023
  2. Conjugates of Tacrine and Salicylic Acid Derivatives as New Promising Multitarget Agents for Alzheimer’s Disease

    Makhaeva, G. F., Kovaleva, N. V., Rudakova, E. V., Boltneva, N. P., Grishchenko, M. V., Lushchekina, S. V., Astakhova, T. Y., Serebryakova, O. G., Timokhina, E. N., Zhilina, E. F., Shchegolkov, E. V., Ulitko, M. V., Radchenko, E. V., Palyulin, V. A., Burgart, Y. V., Saloutin, V. I., Bachurin, S. O. & Richardson, R. J., Jan 2023, In: International Journal of Molecular Sciences. 24, 3, 2285.

    Research output: Contribution to journalArticlepeer-review

  3. Powerful Potential of Polyfluoroalkyl-Containing 4-Arylhydrazinylidenepyrazol-3-ones for Pharmaceuticals

    Burgart, Y. V., Elkina, N. A., Shchegolkov, E. V., Krasnykh, O. P., Makhaeva, G. F., Triandafilova, G. A., Solodnikov, S. Y., Boltneva, N. P., Rudakova, E. V., Kovaleva, N. V., Serebryakova, O. G., Ulitko, M. V., Borisevich, S. S., Gerasimova, N. A., Evstigneeva, N. P., Kozlov, S. A., Korolkova, Y. V., Minin, A. S., Belousova, A. V., Mozhaitsev, E. S., & 2 othersKlabukov, A. M. & Saloutin, V. I., 2023, In: Molecules. 28, 1, 59.

    Research output: Contribution to journalArticlepeer-review

  4. 2022
  5. Synthesis of 4-Aminopyrazol-5-ols as Edaravone Analogs and Their Antioxidant Activity

    Burgart, Y. V., Makhaeva, G. F., Krasnykh, O. P., Borisevich, S. S., Agafonova, N. A., Kovaleva, N. V., Boltneva, N. P., Rudakova, E. V., Shchegolkov, E. V., Triandafilova, G. A., Gazizov, D. A., Serebryakova, O. G., Ulitko, M. V., Khursan, S. L., Saloutin, V. I. & Richardson, R. J., Nov 2022, In: Molecules. 27, 22, 7722.

    Research output: Contribution to journalArticlepeer-review

  6. Promising Antifungal and Antibacterial Agents Based on 5-Aryl-2,2 '-bipyridines and Their Heteroligand Salicylate Metal Complexes: Synthesis, Bioevaluation, Molecular Docking

    Burgart, Y., Shchegolkov, E., Shchur, I., Kopchuk, D., Gerasimova, N., Borisevich, S., Evstigneeva, N., Zyryanov, G., Savchuk, M., Ulitko, M., Zilberberg, N., Kungurov, N., Saloutin, V., Charushin, V. & Chupakhin, O., 4 Feb 2022, In: ChemMedChem. 17, 3, 15 p., e202100577.

    Research output: Contribution to journalArticlepeer-review

  7. 2021
  8. Synthesis of new efficient and selective carboxylesterase inhibitors based on adamantyl and citronellyl 4,4,4-trifluoro-2-arylhydrazonylidene-3-oxobutanoates

    Elkina, N. A., Shchegolkov, E. V., Burgart, Y. V., Saloutin, V. I., Boltneva, N. P., Serebryakova, O. G., Lushchekina, S. V. & Makhaeva, G. F., Mar 2021, In: Russian Chemical Bulletin. 70, 3, p. 567-572 6 p.

    Research output: Contribution to journalArticlepeer-review

  9. Copper(II) and cobalt(II) complexes based on methyl trifluorosalicylate and bipyridine-type ligands: Synthesis and their antimicrobial activity

    Shchegolkov, E. V., Shchur, I. V., Burgart, Y. V., Slepukhin, P. A., Evstigneeva, N. P., Gerasimova, N. A., Zilberberg, N. V., Kungurov, N. V., Saloutin, V. I. & Chupakhin, O. N., 15 Jan 2021, In: Polyhedron. 194, 10 p., 114900.

    Research output: Contribution to journalArticlepeer-review

  10. СИНТЕЗ НОВЫХ ЭФФЕКТИВНЫХ И СЕЛЕКТИВНЫХ ИНГИБИТОРОВ КАРБОКСИЛЭСТЕРАЗЫ НА ОСНОВЕ АДАМАНТИЛИ ЦИТРОНЕЛЛИЛ-4,4,4-ТРИФТОР-2-АРИЛГИДРАЗИНИЛИДЕН-3-ОКСОБУТАНОАТОВ

    Елькина, Н. А., Щегольков, Е. В., Бургарт, Я. В., Салоутин, В. И., Болтнева, Н. П., Серебрякова, О. Г., Лущекина, С. В. & Махаева, Г. Ф., 2021, In: Известия Академии наук. Серия химическая. 3, p. 567-572 6 p.

    Research output: Contribution to journalArticlepeer-review

  11. 2020
  12. Multiple biological active 4-aminopyrazoles containing trifluoromethyl and their 4-nitroso-precursors: Synthesis and evaluation

    Burgart, Y. V., Agafonova, N. A., Shchegolkov, E. V., Krasnykh, O. P., Kushch, S. O., Evstigneeva, N. P., Gerasimova, N. A., Maslova, V. V., Triandafilova, G. A., Solodnikov, S. Y., Ulitko, M. V., Makhaeva, G. F., Rudakova, E. V., Borisevich, S. S., Zilberberg, N. V., Kungurov, N. V., Saloutin, V. I. & Chupakhin, O. N., 15 Dec 2020, In: European Journal of Medicinal Chemistry. 208, 17 p., 112768.

    Research output: Contribution to journalArticlepeer-review

  13. Competitive routes to cyclizations of polyfluoroalkyl-containing 2-tolylhydrazinylidene-1,3-diketones with 3-aminopyrazoles into bioactive pyrazoloazines

    Elkina, N. A., Burgart, Y. V., Shchegolkov, E. V., Krasnykh, O. P., Maslova, V. V., Triandafilova, G. A., Solodnikov, S. S., Muryleva, A. A., Misiurina, M. A., Slita, A. V., Zarubaev, V. V. & Saloutin, V. I., Dec 2020, In: Journal of Fluorine Chemistry. 240, 11 p., 109648.

    Research output: Contribution to journalArticlepeer-review

  14. Synthesis and biological activity of polyfluorinated p-aminosalicylic acids and their amides

    Burgart, Y. V., Shchur, I. V., Shchegolkov, E. V. & Saloutin, V. I., 1 Sept 2020, In: Mendeleev Communications. 30, 5, p. 636-638 3 p.

    Research output: Contribution to journalArticlepeer-review

Previous 1 2 3 Next

ID: 7874490